Potential Anticancer Agents.1 LXII. The Relationship of Chemical Structure to Antileukem'c Activity with Analogs of 1-Methyl-3-nitro-1-nitrosoguanidine (NSC-9369). II Karen A. Hyde, Edward Acton, W. A. Skinner, Leon Goodman, Joseph Greenberg, and B. R. Baker pp 1 - 14; DOI: 10.1021/jm01236a001 |
Synthesis of Potential Anticancer Agents. XXX. (1-Aziridinyl)purines J. A. Montgomery, K. Hewson, and C. Temple pp 15 - 24; DOI: 10.1021/jm01236a002 |
Complex Esters of Thioinosinic-(5′) Acid H. Jeanette Thomas and John A. Montgomery pp 24 - 32; DOI: 10.1021/jm01236a003 |
para-[N-Bis-(2-chloroethyl)]-aminobenzoylglutamic Acid S.-C. J. Fu pp 33 - 41; DOI: 10.1021/jm01236a004 |
Synthesis of Peptides of 1-Aminocyclopentanecarboxylic Acid S. Shankman, S. Higa, F. Lew, and M. E. Roberts pp 42 - 49; DOI: 10.1021/jm01236a005 |
Pyridoxal Hydrazine Derivatives for Cancer Chemotherapy Richard H. Wiley and Gether Irick pp 49 - 53; DOI: 10.1021/jm01236a006 |
2-tert-Butyl-10-(3-dimethylaminopropyl)-phenothiazine and Related Compounds Francis Sowinski and Harry L. Yale pp 54 - 63; DOI: 10.1021/jm01236a007 |
Some Analogs of Chlordiazepoxide S. C. Bell, C. Gochman, and S. J. Childress pp 63 - 69; DOI: 10.1021/jm01236a008 |
Indanols. IV.1 Indanoxypropanolamines Seymour L. Shapiro, Vincent A. Parrino, Elaine S. Isaacs, and Louis Freedman pp 69 - 76; DOI: 10.1021/jm01236a009 |
α-Benzyltetrahydrofurfurylamines--a New Series of Psychomotor Stimulants. I Robert L. Clarke and Louis S. Harris pp 77 - 95; DOI: 10.1021/jm01236a010 |
Hypotensive Agents. 2-(2-Aminoethyl)-piperidine Derivatives William F. Minor, Justin B. Hoekstra, Dorothea Fisher, and Joseph Sam pp 96 - 107; DOI: 10.1021/jm01236a011 |
16-Substituted Steroids. XVIII.1 6,16-Difunctional 3,5-Cyclo-5α-androstanes James R. Rhone, Max N. Huffman, and Allan J. Stanley pp 107 - 111; DOI: 10.1021/jm01236a012 |
The Solvolysis of 21-Hydrocortisone Esters and Hemiesters Edward R. Garrett pp 112 - 133; DOI: 10.1021/jm01236a013 |
Certain Steroid Ketals and Their Biological Activity William S. Allen, Henry M. Kissman, Sidney Mauer, Ira Ringler, and Martin J. Weiss pp 133 - 155; DOI: 10.1021/jm01236a014 |
Mercury Derivatives of Allylhydantoins Franklyn W. Gubitz and William B. McKeon pp 168 - 175; DOI: 10.1021/jm01236a015 |
Potential Uricosuric Agents Derived from 1,3-Diphenylbarbituric Acid Homer C. Scarborough and Gordon R. McKinney pp 175 - 183; DOI: 10.1021/jm01236a016 |
Large Scale Preparation and Purification of the Vasopressor Polypeptide, Substance A C. G. Huggins and E. J. Walaszek pp 183 - 190; DOI: 10.1021/jm01236a017 |
Penetration of Brain and Brain Tumor by Aromatic Compounds as a Function of Molecular Substituents. III A. H. Soloway, B. Whitman, and J. R. Messer pp 191 - 196; DOI: 10.1021/jm01236a018 |
Aspects of the Metabolism of Isoniazid and Acetylisoniazid in the Human and the Dog Allen S. Yard and Herbert McKennis pp 196 - 203; DOI: 10.1021/jm01236a019 |
A Metabolic Study of α-Methyl-β-(3,4-dihydroxyphenyl)-DL-alanine in Man Theodore L. Sourkes, Gerard F. Murphy, and Beatriz Chavez-Lara pp 204 - 210; DOI: 10.1021/jm01236a020 |
Comparison between the Rate Constants for Acetylation of Sulfonamides in Vivo and O/W Partition Coefficient Eino Nelson pp 211 - 214; DOI: 10.1021/jm01236a021 |
The Mechanism of Action of the 2-Phenylcyclopropylamine Type of Monoamine Oxidase Inhibitors B. Belleau and J. Moran pp 215 - 219; DOI: 10.1021/jm01236a022 |
Book Review pp 220 - 220; DOI: 10.1021/jm01236a023 |
Synthesis of Sulfonylhydrazine Derivatives with Monoamine Oxidase Inhibitory Activity C. S. Rooney, Edward J. Cragoe, Jr, Curt C. Porter, and James M. Sprague pp 155 - 167; DOI: 10.1021/jm01236a600 |
Chemistry and Pharmacology of Monoamine Oxidase Inhibitors: Hydrazine Derivatives Floyd E. Anderson, Daniel Kaminsky, Bernard Dubnick, Sylvester R. Klutchko, Wiaczeslaw A. Cetenko, Jonas Gylys, and John A. Hart pp 221 - 230; DOI: 10.1021/jm01237a001 |
Hypoglycemic Activity in Relation to Chemical Structure of Potential Oral Antidiabetic Substances. I. 1-Sulfonyl-3-alkylureas Bernt Hökfelt and Åke Jönsson pp 231 - 239; DOI: 10.1021/jm01237a002 |
Hypoglycemic Activity in Relation to Chemical Structure of Potential Oral Antidiabetic Substances. II. Analogs of 1-Sulfonyl-3-alkylureas Bernt Hökfelt and Åke Jönsson pp 240 - 246; DOI: 10.1021/jm01237a003 |
Hypoglycemic Activity in Relation to Chemical Structure of Potential Oral Antidiabetic Substances. III. 2-Benzenesulfonamido-5-alkyl-1,3,4-thiadiazoles and -oxadiazoles Bernt Hökfelt and Åke Jönsson pp 247 - 257; DOI: 10.1021/jm01237a004 |
Dihydro-1,3-oxazines as Antitumor Agents M. E. Kuehne and E. A. Konopka pp 257 - 280; DOI: 10.1021/jm01237a005 |
Steroidal Dihydro-1,3-oxazines as Antitumor Agents M. E. Kuehne, E. A. Konopka, and B. F. Lambert pp 281 - 296; DOI: 10.1021/jm01237a006 |
Antineoplastic Agents. IV. Mannich Base Nitrogen Mustards (Part A)1,2,3 George R. Pettit and Joseph A. Settepani pp 296 - 302; DOI: 10.1021/jm01237a007 |
6-Acylamido- and 6-Acylamido-9(or 7)-acylpurines Arnold H. Schein pp 302 - 311; DOI: 10.1021/jm01237a008 |
Structure-Activity Relationships of 3-Substituted Dihydrobenzothiadiazine Diuretics Richard M. Taylor and John G. Topliss pp 312 - 320; DOI: 10.1021/jm01237a009 |
Coumestrol, Plant Phenolics, and Synthetic Estrogens: a Correlation of Structure and Activity Robert A. Micheli, A. N. Booth, A. L. Livingston, and E. M. Bickoff pp 321 - 335; DOI: 10.1021/jm01237a010 |
Oxazolocoumarins Robert Bruce Moffett pp 335 - 340; DOI: 10.1021/jm01237a011 |
3-Substituted Tropane Derivatives. III. 3-Substituted Tropane Carbinols, Alkenes, and Alkanes Charles L. Zirkle, Elvin L. Anderson, Paul N. Craig, Fred R. Gerns, Zena K. Indik, and Alex M. Pavloff pp 341 - 356; DOI: 10.1021/jm01237a012 |
Structures Related to Morphine. XXII.1 A Benzomorphan Congener of Meperidine Hiroshi Kugita, Seiichi Saito, and Everette L. May pp 357 - 361; DOI: 10.1021/jm01237a013 |
α-Benzyltetrahydrofurfurylamines--A New Series of Psychomotor Stimulants. II.1 Resolution of Isomers Robert L. Clarke, B. F. Tullar, and Louis S. Harris pp 362 - 372; DOI: 10.1021/jm01237a014 |
Dialkylaminoalkyl Derivatives of 10,11-Dihydro-5H-dibenzo[a,d]cycloheptene and Related Compounds Frank J. Villani, Claire A. Ellis, Carol Teichman, and Catherine Bigos pp 373 - 383; DOI: 10.1021/jm01237a015 |
The Anticonvulsant Activity of 1,2,4-Triazoles C. Ainsworth, Nelson R. Easton, M. Livezey, D. E. Morrison, and W. R. Gibson pp 383 - 389; DOI: 10.1021/jm01237a016 |
Derivatives of 8-Hydroxy-2-quinolineacrylic Acid. II Madhukar G. Vaidya and Joseph G. Cannon pp 389 - 397; DOI: 10.1021/jm01237a017 |
Synthesis of Potential Anticancer Agents. VII. Some 3-Chloropropionyl Amides1-3 Frank D. Popp, Ernest Cullen, Robert B. Davis, and Warren Kirsch pp 398 - 403; DOI: 10.1021/jm01237a018 |
An Improved Procedure for Preparing 1-Methylpyridinium-2-aldoxime Chloride Robert I. Ellin, David Easterday, and Albert A. Kondritzer pp 404 - 405; DOI: 10.1021/jm01237a019 |
Steroids. CLXXX.1 2-Methyl-Δ2-androstenes and 2-Methylene-androstanes. A New Class of Potent Anabolic Agents A. D. Cross, J. A. Edwards, and A. Bowers pp 406 - 408; DOI: 10.1021/jm01237a020 |
Steroids. CLXXXIV.1 2-Formyl-Δ2-androstenes and Related Compounds. A New Class of Potent Anabolic Agents J. C. Orr, O. Halpern, and A. Bowers pp 409 - 411; DOI: 10.1021/jm01237a021 |
Book Review pp 412 - 412; DOI: 10.1021/jm01237a022 |
Synthesis and Biological Properties of 9-Sarcosine Oxytocin William D. Cash, Logan McCulloch Mahaffey, Alfred S. Buck, Donald E. Nettleton, Christos Romas, and Vincent du Vigneaud pp 413 - 423; DOI: 10.1021/jm01238a001 |
Isomeric 2-Acetoxytropine Methiodides S. Archer, A. M. Lands, and T. R. Lewis pp 423 - 430; DOI: 10.1021/jm01238a002 |
Synthesis and Analgesic Activity of a New Bridged Heterocyclic System H. E. Zaugg, R. W. DeNet, and E. T. Kimura pp 430 - 440; DOI: 10.1021/jm01238a003 |
Analgetics Based on the Pyrrolidine Ring. II. J. F. Cavalla, R. A. Selway, J. Wax, L. Scotti, and C. V. Winder pp 441 - 451; DOI: 10.1021/jm01238a004 |
Structure-Activity Relationships in a Series of Anticonvulsant and Hypnotic Bicyclic Carboxamides Werner R. Boehme, Estelle A. Siegmund, William G. Scharpf, and Edgar Schipper pp 451 - 464; DOI: 10.1021/jm01238a005 |
The Synthesis and γ-Aminobutyric Acid Transaminase Inhibition of Aminoöxy Acids and Related Compounds E. L. Schumann, L. A. Paquette, R. V. Heinzelman, D. P. Wallach, J. P. DaVanzo, and M. E. Greig pp 464 - 477; DOI: 10.1021/jm01238a006 |
Anabolic Agents: Derivatives of 2-Halo-5α-androst-1-ene R. E. Counsell and P. D. Klimstra pp 477 - 483; DOI: 10.1021/jm01238a007 |
The Metabolites of Ergometrine and Lysergic Acid Diethylamide in Rat Bile M. B. Slaytor and S. E. Wright pp 483 - 491; DOI: 10.1021/jm01238a008 |
The Fate and Excretion of Polythiazide1 in the Dog Rex Pinson, Eric C. Schreiber, Edward H. Wiseman, Josephine Chiaini, and Doris Baumgartner pp 491 - 503; DOI: 10.1021/jm01238a009 |
Monoamine Oxidase Inhibitors. III. Structural Variations in 1-Alkyl and 1-Aralkyl-1(or 2)-acylhydrazines Thomas S. Gardner, Edward Wenis, and John Lee pp 503 - 513; DOI: 10.1021/jm01238a010 |
Reduction of Nitrofurans. I. Aminofurans Frank F. Ebetino, James J. Carroll, and Gabriel Gever pp 513 - 524; DOI: 10.1021/jm01238a011 |
The Metabolism of 5-Nitro-2-furaldehyde Acetylhydrazone Joanne Olivard, Salvatore Valenti, and James A. Buzard pp 524 - 531; DOI: 10.1021/jm01238a012 |
Synthesis and Biological Activity of Pyridoxine Analogs Shreekrishna M. Gadekar, Jean L. Frederick, and Edward C. DeRenzo pp 531 - 538; DOI: 10.1021/jm01238a013 |
6-Deoxytetracyclines. II. Nitrations and Subsequent Reactions J. Petisi, J. L. Spencer, J. J. Hlavka, and J. H. Boothe pp 538 - 546; DOI: 10.1021/jm01238a014 |
Synthetic Amebicides. VI. Benzo[b][1,8]phenanthrolines, Benzo[b][1,10]phenanthrolines, Dibenzo[b,h][1,6]naphthyridines, and Benzo[h]quino[4,3-b]quinolines Edward F. Elslager and Frank H. Tendick pp 546 - 558; DOI: 10.1021/jm01238a015 |
Potential Purine Antagonists. XXXI. The Preparation of Certain 9-Alkyl-2-amino-6-purinethiols and Related Derivatives as Antitumor Agents C. Wayne Noell and Roland K. Robins pp 558 - 588; DOI: 10.1021/jm01238a016 |
Potential Purine Antagonists. XXXII. The Synthesis and Antitumor Activity of Certain Compounds Related to 4-Aminopyrazolo[3,4-d]pyrimidine Edward Y. Sutcliffe, K. Y. Zee-Cheng, C. C. Cheng, and Roland K. Robins pp 588 - 607; DOI: 10.1021/jm01238a017 |
The Preparation and Antitumor Activity of Certain Derivatives of 6-Mercaptopurine Leland R. Lewis, C. Wayne Noell, Alden G. Beaman, and Roland K. Robins pp 607 - 617; DOI: 10.1021/jm01238a018 |
Potential Hypoglycemic Agents: 1,3,4-Oxadiazoles and Related Compounds J. B. O'Neal, H. Rosen, P. B. Russell, A. C. Adams, and A. Blumenthal pp 617 - 626; DOI: 10.1021/jm01238a019 |
Synthesis of Potential Anticancer Agents. VIII. Benzaldehyde Mustard Derivatives and Related Compounds Frank D. Popp pp 627 - 629; DOI: 10.1021/jm01238a020 |
Microbiological Transformation of Strophanthidin Charles J. Sih, S. Morris Kupchan, O. El Tayeb, and Adriano Afonso pp 629 - 633; DOI: 10.1021/jm01238a021 |
New Benzomorphan Analgetics Maxwell Gordon, John J. Lafferty, David H. Tedeschi, Blaine M. Sutton, Nathan B. Eddy, and Everett L. May pp 633 - 635; DOI: 10.1021/jm01238a022 |
Blockade of Adrenergic α-Receptors by a Carbonium Ion B. Belleau and D. J. Triggle pp 636 - 639; DOI: 10.1021/jm01238a023 |
Pyrimidines. VIII. Pyrimidine Derivatives of Thioguanine H. C. Koppel, Robert Henre Springer, Roland K. Robins, and C. C. Cheng pp 639 - 641; DOI: 10.1021/jm01238a024 |
Intestinal Anthelmintics. I. The Preparation of Bis(2,4,5-trichlorophenol)-Piperazine Salt (Triclofenol Piperazine) and Other Phenol-Piperazine Salts Franklin W. Short and Edward F. Elslager pp 642 - 646; DOI: 10.1021/jm01238a025 |
Synthetic Amebicides. VII. 6,6′-Diallyl-α,α′-bis(dialkylaminoalkylamino)-4,4′-bi-o -cresols Edward F. Elslager and Frank H. Tendick pp 646 - 651; DOI: 10.1021/jm01238a026 |
Preparation of Amidines by Catalytic Reduction of Amidoximes Robert P. Mull, Renat H. Mizzoni, Mary R. Dapero, and Mary E. Egbert pp 651 - 654; DOI: 10.1021/jm01238a027 |
Non-classical Antimetabolites. VII.1,2 The Bridge Principle of Specificity with Exo-alkylating Irreversible Inhibitors B. R. Baker pp 654 - 656; DOI: 10.1021/jm01238a028 |
Tumor Inhibitors. I. Aristolochic Acid, the Active Principle of Aristolochia indica S. Morris Kupchan and Raymond W. Doskotch pp 657 - 659; DOI: 10.1021/jm01238a029 |
α,β-Unsaturated Ketone Derivatives of Aryloxyacetic Acids, a New Class of Diuretics Everett M. Schultz, Edward J. Cragoe, John B. Bicking, William A. Bolhofer, and James M. Sprague pp 660 - 662; DOI: 10.1021/jm01238a030 |
Book Reviews pp 663 - 664; DOI: 10.1021/jm01238a031 |
Chemistry and Structure-Activity Relationships of Mecamylamine and Derivatives Clement A. Stone, Mary L. Torchiana, Katherine L. Meckelnberg, John Stavorski, Meyer Sletzinger, Gustav A. Stein, William V. Ruyle, Donald F. Reinhold, Walter A. Gaines, Heinz Arnold, and Karl Pfister pp 665 - 690; DOI: 10.1021/jm01239a001 |
Veratrum Alkaloids. XLIX.1 The Structures and Configurations of Sabine and Sabadine2,3 S. Morris Kupchan, Norbert Gruenfeld, and N. Katsui pp 690 - 714; DOI: 10.1021/jm01239a002 |
Degradation of Corticosteroids. VII. The Synthesis of 7-Membered Ring-A Enol-Lactones E. Caspi, Y. W. Chang, and R. I. Dorfman pp 714 - 719; DOI: 10.1021/jm01239a003 |
Hypocholesterolemic Agents. I. 20α-(2-Dialkylaminoethyl)aminopregn-5-en-3β-ol Derivatives R. E. Counsell, P. D. Klimstra, R. E. Ranney, and D. L. Cook pp 720 - 729; DOI: 10.1021/jm01239a004 |
Thyroxine Analogs. VI.1 Synthesis and Antigoitrogenic Activity of 3,5-Diiodo-4-(4′-Aminophenoxy)-L-Phenylalanines, Including the 4′-Amino Analog of 3,5,3′-Triiodo-L-Thyronine Eugene C. Jorgensen and Peter Slade pp 729 - 738; DOI: 10.1021/jm01239a005 |
Studies on Monoamine Oxidase Inhibitors. I. The Autoxidation of β-Phenylisopropylhydrazine as a Model Reaction for Irreversible Monoamine Oxidase Inhibition L. E. Eberson and K. Persson pp 738 - 752; DOI: 10.1021/jm01239a006 |
Pyrrolidines. VII. 3-Hydroxy-1-Pyrrolidinecarboxylic Acid Esters Yao-Hua Wu, William A. Gould, Walter G. Lobeck, Herbert R. Roth, and R. F. Feldkamp pp 752 - 762; DOI: 10.1021/jm01239a007 |
Pyrrolidines. VIII. 3-Acyloxy-3-Aryl-1-Ethyl-and -1-Methylpyrrolidines Yao-Hua Wu, Walter G. Lobeck, and R. F. Feldkamp pp 762 - 769; DOI: 10.1021/jm01239a008 |
Structure-Activity Relationships in a Series of Anticonvulsant Bicyclic Acylureas Werner R. Boehme, Estelle A. Siegmund, William G. Scharpf, and Edgar Schipper pp 769 - 775; DOI: 10.1021/jm01239a009 |
Some Aspects of the Chemistry of 5-Ethyl-6-phenyl-meta-thiazane-2,4-dione, an Anesthetic Agent Robert G. Taborsky and Roland J. Starkey pp 775 - 780; DOI: 10.1021/jm01239a010 |
Acetylenic Amines. III. The Haloethynyl Derivatives C. W. Ryan, Nelson R. Easton, Robert D. Dillard, and Francis G. Henderson pp 780 - 784; DOI: 10.1021/jm01239a011 |
Synthesis and Hypotensive Activity of Unsymmetrically Substituted Acetylenic Bis-Quaternary Ammonium Compounds and Certain of Their Reduction Products John L. Neumeyer, Joseph G. Cannon, and Joseph P. Buckley pp 784 - 792; DOI: 10.1021/jm01239a012 |
Apparent Dissociation Constants of Haloaralkylamines Seymour L. Shapiro, Elaine S. Isaacs, Victor Bandurco, and Louis Freedman pp 793 - 799; DOI: 10.1021/jm01239a013 |
Antineoplastic Agents. V. The Aromatic System of Podophyllotoxin (Part B)1-3 George R. Pettit, Michael F. Baumann, and K. N. Rangammal pp 800 - 808; DOI: 10.1021/jm01239a014 |
The Syntheses and Pharmacological Activities of Amide, Sulfamide, and Urea Derivatives of 4,6-Diaminopyrimidines John J. Traverso, E. Brown Robbins, and Calvert W. Whitehead pp 808 - 815; DOI: 10.1021/jm01239a015 |
Antidiabetic Agents. N4-Arylsulfonylsemicarbazides John B. Wright and Robert E. Willette pp 815 - 822; DOI: 10.1021/jm01239a016 |
Antituberculous Agents. II.1 N,N′-Diisopropylethylenediamine and Analogs R. G. Shepherd and R. G. Wilkinson pp 823 - 835; DOI: 10.1021/jm01239a017 |
Antituberculous Agents. III. (+)-2,2 -(Ethylenediimino)-di-1-butanol1,2 and Some Analogs R. G. Wilkinson, M. B. Cantrall, and R. G. Shepherd pp 835 - 845; DOI: 10.1021/jm01239a018 |
Antiradiation Compounds. II. Dithiocarbamates William O. Foye and James Mickles pp 846 - 852; DOI: 10.1021/jm01239a019 |
Synthesis of Chromogenic Substrates for the Assay of Aminopeptidase Activity Theodore P. Goldstein, Robert E. Plapinger, Marvin M. Nachlas, and Arnold M. Seligman pp 852 - 857; DOI: 10.1021/jm01239a020 |
The Biological Activity of Certain 17α,20; 20,21-Bismethylenedioxy Corticoid Derivatives Martin J. Weiss, Robert E. Schaub, and Sidney Mauer pp 858 - 861; DOI: 10.1021/jm01239a021 |
Synthesis of Sydnones and Sydnone Imines Claude V. Greco, Wayne H. Nyberg, and C. C. Cheng pp 861 - 865; DOI: 10.1021/jm01239a022 |
Synthesis of Potential Antineoplastic Agents. XXXI. 9-Alkyl-9H-Purines Carroll Temple, Conrad L. Kussner, and John A. Montgomery pp 866 - 870; DOI: 10.1021/jm01239a023 |
Synthesis and Biological Activity of Some 4-(Substituted)aminopyrimidines Hayim Segal, Charles Hedgcoth, and Charles G. Skinner pp 871 - 876; DOI: 10.1021/jm01239a024 |
C(19)-Substituted Steroid Hormone Analogs. I. 17β-Hydroxy-3-oxoandrost-4-ene-19-nitrile Timothy Jen and Manfred E. Wolff pp 876 - 878; DOI: 10.1021/jm01239a025 |
Book Reviews pp 879 - 882; DOI: 10.1021/jm01239a026 |
Bicyclic Bases. IV.1 Aryl Substituted Bridged Hydroisoindolines George I. Poos, Margaret M. Lehman, Elizabeth B. Landis, and Janet D. Rosenau pp 883 - 896; DOI: 10.1021/jm01240a001 |
Synthesis and Diuretic Activity of 3,3-Spiro-Substituted Hydrothiazides Edward J. Cragoe, Otto W. Woltersdorf, John E. Baer, and James M. Sprague pp 896 - 912; DOI: 10.1021/jm01240a002 |
Strong Analgesics. Some 1-Substituted 4-Phenyl-4-Propionoxypiperidines Philip M. Carabateas and Leonard Grumbach pp 913 - 919; DOI: 10.1021/jm01240a003 |
Dicarbamates and Thiolcarbamates George deStevens, Marylou Sklar, Halina Lukaszewski, and Lloyd Witkin pp 919 - 924; DOI: 10.1021/jm01240a004 |
Structure-Activity Relationships of Ethylenimines. II. Methyl-Substituted Derivatives of Tetramin Albert T. Bottini and Vasu Dev pp 925 - 932; DOI: 10.1021/jm01240a005 |
Structure-Activity Relationships of 1-[3-Indolyl)alkyl]-4-arylpiperazines. A New Series of Tranquilizers David W. Wylie and S. Archer pp 932 - 943; DOI: 10.1021/jm01240a006 |
Guanidines with Antihypertensive Activity. II Robert P. Mull, Renat H. Mizzoni, Mary R. Dapero, and Mary E. Egbert pp 944 - 949; DOI: 10.1021/jm01240a007 |
Synthesis of Certain C-2 and C-6 Substituted Derivatives of 9α-Fluoro-16α-hydroxyhydrocortisone 16,17-Acetonide Henry M. Kissman, Arlene Small Hoffman, John F. Poletto, and Martin J. Weiss pp 950 - 962; DOI: 10.1021/jm01240a008 |
Synthesis of Certain 16α-Substituted Derivatives of 9α-Fluoro-11-dehydrocorticosterone, Progesterone and Deoxycorticosterone Arlene Small Hoffman, Henry M. Kissman, and Martin J. Weiss pp 962 - 975; DOI: 10.1021/jm01240a009 |
16-Alkylated Progesterones Elliot Shapiro, Theodore Legatt, Lois Weber, Merl Steinberg, A. Watnick, M. Eisler, Marilyn Gilmore Hennessey, C. T. Coniglio, W. Charney, and Eugene P. Oliveto pp 975 - 988; DOI: 10.1021/jm01240a010 |
Cardiac Activity of Newer Digitalis Glycosides and Aglycones Francis G. Henderson and K. K. Chen pp 988 - 995; DOI: 10.1021/jm01240a011 |
Synthesis and Antitumor Activity of 2-Amino-1-methylpurine-6-thione C. Wayne Noell, Donald W. Smith, and Ronald K. Robins pp 996 - 999; DOI: 10.1021/jm01240a012 |
Synthesis of Potential “Dual Antagonists.” I. Some Bis(1-aziridinyl)phosphinyl Carbamates1 and Their Structural Analogs Zinon B. Papanastassiou and Thomas J. Bardos pp 1000 - 1007; DOI: 10.1021/jm01240a013 |
Synthesis of Compounds Related to 2-(o-chlorophenyl)-2-(p-chlorophenyl)-1,1-dichloroethanea Kwang Yuen Zee-Cheng and C. C. Cheng pp 1008 - 1015; DOI: 10.1021/jm01240a014 |
Derivatives of 6-Aminopenicillanic Acid. III. Reactions with N-Substituted Phthalamic Acids Y. G. Perron, W. F. Minor, L. B. Crast, A. Gourevitch, J. Lein, and L. C. Cheney pp 1016 - 1025; DOI: 10.1021/jm01240a015 |
N(α-D-Penicilloyl) Amines as Univalent Hapten Inhibitors of Antibody-Dependent Allergic Reactions to Penicillin Bernard B. Levine pp 1025 - 1034; DOI: 10.1021/jm01240a016 |
In vitro Metabolism of 2-Chloro-10-(3-dimethylaminopropyl)-phenothiazine. III. Isolation and Identification of Metabolites John J. Ross, Thomas L. Flanagan, and Alfred R. Maass pp 1035 - 1041; DOI: 10.1021/jm01240a017 |
Chemotherapeutic Nitrofurans. VIII.1 The Synthesis of Certain 3,4-Dichloro-5-nitrofurans Julian G. Michels, Gabriel Gever, and Peter H. L. Wei pp 1042 - 1048; DOI: 10.1021/jm01240a018 |
Disubstituted Progesterones. The 6,16-Chloro and Methyl Series Richard T. Rapala and Mauriec J. Murray pp 1049 - 1053; DOI: 10.1021/jm01240a019 |
Some New Synthetic Flavonoid Glycosides Related in Structure to Phlorizin Donald F. Diedrich pp 1054 - 1062; DOI: 10.1021/jm01240a020 |
1,8-Naphthyridine Derivatives. A New Class of Chemotherapeutic Agents George Y. Lesher, Ernest J. Froelich, Monte D. Gruett, John Hays Bailey, and R. Pauline Brundage pp 1063 - 1065; DOI: 10.1021/jm01240a021 |
Book Reviews pp 1066 - 1066; DOI: 10.1021/jm01240a022 |
The Synthesis of 6-Fluoro-9-methylpurine Alden G. Beaman and Roland K. Robins pp 1067 - 1074; DOI: 10.1021/jm01241a001 |
The Antitumor Activity of 2-Amino-6-alkylthio-9-(β-D-ribofuranosylpurines and related Derivatives of 2-Amino-6-purinethiol (Thioguanine) C. Wayne Noell and Roland K. Robins pp 1074 - 1085; DOI: 10.1021/jm01241a002 |
Pyrimidines. IX. 4- and 5-(Substituted-anilino)pyrimidines Darrell E. O'Brien, Fred Baiocchi, Roland K. Robins, and C. C. Cheng pp 1085 - 1103; DOI: 10.1021/jm01241a003 |
5-Benzyl-2,4-diaminopyrimidines as Antibacterial Agents. I. Synthesis and Antibacterial Activity in vitro Barbara Roth, Elvira A. Falco, George H. Hitchings, and S. R. M. Bushby pp 1103 - 1123; DOI: 10.1021/jm01241a004 |
Synthesis of Aminosugar Nucleosides Calvin L. Stevens and K. Nagarajan pp 1124 - 1148; DOI: 10.1021/jm01241a005 |
9-Amino-2,3-dimethoxy-6-nitroacridine 10-Oxides Edward F. Elslager and Frank H. Tendick pp 1149 - 1153; DOI: 10.1021/jm01241a006 |
4-(3-Chloro-9-acridinylamino)-α-amino-o-cresol 10-Oxides Edward F. Elslager and Frank H. Tendick pp 1153 - 1158; DOI: 10.1021/jm01241a007 |
3-Chloro-9-(4-diethylamino-1-methylbutylamino)acridine 10-Oxide and other 9-Aminoacridine N-Oxides Edward F. Elslager, Ralph E. Bowman, Frank H. Tendick, David J. Tivey, and Donald F. Worth pp 1159 - 1176; DOI: 10.1021/jm01241a008 |
Mono- and Difluorination of Steroids at C-16 through Enamine Intermediates Arthur H. Goldkamp pp 1176 - 1187; DOI: 10.1021/jm01241a009 |
The Synthesis of Some Acidic Amino Acids Possessing Neuropharmacological Activity J. C. Watkins pp 1187 - 1199; DOI: 10.1021/jm01241a010 |
New Psychotropic Agents.1 II. Derivatives of 5,6-Dihydrodibenz[b,e]azepine (5,6-Dihydromorphanthridine) Stanley O. Winthrop, M. A. Davis, F. Herr, J. Stewart, and Roger Gaudry pp 1199 - 1206; DOI: 10.1021/jm01241a011 |
New Psychotropic Agents.1 III. Derivatives of 6,11-Dihydrodibenz[b,e]oxepine and 6,11-Dihydrodibenzo[b,e]thiepine Stanley O. Winthrop, M. A. Davis, F. Herr, J. Stewart, and Roger Gaudry pp 1207 - 1215; DOI: 10.1021/jm01241a012 |
Hypocholesterolemic Agents. II.1 2β-Halo-5α-androstane Derivatives P. D. Klimstra and R. E. Counsell pp 1216 - 1224; DOI: 10.1021/jm01241a013 |
Hypocholesterolemic Agents. III.1 N-Methyl-N-(dialkylamino)alkyl-17β-aminoandrost-5-en-3β-ol Derivatives R. E. Counsell, P. D. Klimstra, and R. E. Ranney pp 1224 - 1233; DOI: 10.1021/jm01241a014 |
A Chemical and Pharmacological Study of Some Compounds Derived from 3,4-Xylidine Dinah M. James and Alun H. Rees pp 1234 - 1238; DOI: 10.1021/jm01241a015 |
5-Isonitrosorhodanines Frances C. Brown, Constance M. Harris, and Frances Perry pp 1239 - 1243; DOI: 10.1021/jm01241a016 |
2-Substituted Cyclopropylamines. I. Derivatives and Analogs of 2-Phenylcyclopropylamine Carl Kaiser, Bruce M. Lester, Charles L. Zirkle, Alfred Burger, Charles S. Davis, Thomas J. Delia, and Ludwig Zirngibl pp 1243 - 1265; DOI: 10.1021/jm01241a017 |
2-Substituted Cyclopropylamines. II. Effect of Structure upon Monoamine Oxidase-Inhibitory Activity as Measured in Vivo by Potentiation of Tryptamine Convulsions Charles L. Zirkle, Carl Kaiser, David H. Tedeschi, Ralph E. Tedeschi, and Alfred Burger pp 1265 - 1284; DOI: 10.1021/jm01241a018 |
Researches in the Series of 1,4-Benzodioxane. XXIV. Synthesis and Pharmacological Properties of Some 2-(1-Aminoethyl)-1,4-benzodioxanes D. Misiti, F. De Marchi, V. Rosnati, and D. Bovet pp 1285 - 1293; DOI: 10.1021/jm01241a019 |
The Effect of Methoxyphenyl Substitutions on the Strychnine-Like Activity of Aryldiazaadamantanones and Aryldiazaadamantanols S. Chiavarelli, L. V. Fennoy, G. Settimj, and Leonor De Baran pp 1293 - 1297; DOI: 10.1021/jm01241a020 |
Selective Adrenal Cortical and Gonadal Inhibitors W. L. Bencze and L. I. Barsky pp 1298 - 1306; DOI: 10.1021/jm01241a021 |
Thyroxine Analogs. VIII.1 3-Methyl- and 3,5-Dimethyl-DL-thyronines and Iodinated Derivatives Eugene C. Jorgensen and Robert A. Wiley pp 1307 - 1315; DOI: 10.1021/jm01241a022 |
A Study of the Reaction of the Ascorbic-Dehydroascorbic Acid System and Related Model Compounds with Amphetamine Harold R. Nace and Kenneth F. King pp 1316 - 1327; DOI: 10.1021/jm01241a023 |
Acetylhydrazine as an Intermediate in the Metabolism of Aroylhydrazines Lennox B. Turnbull, Allan S. Yard, and Herbert McKennis pp 1327 - 1334; DOI: 10.1021/jm01241a024 |
Sulfanilamidopyrimidines. II.1 4-Sulfanilamidopyrimidines and Certain 4,6-Disubstituted Pyrimidines2 W. E. Taft and R. G. Shepherd pp 1335 - 1341; DOI: 10.1021/jm01241a025 |
Toxic Constituents of Rayless Goldenrod L. H. Zalkow, N. Burke, G. Cabat, and E. A. Grula pp 1342 - 1351; DOI: 10.1021/jm01241a026 |
Steroids. CLXXV. Further Steroidal Anabolic Agents P. G. Holton and E. Necoechea pp 1352 - 1357; DOI: 10.1021/jm01241a027 |
Spasmolytic 1,2,5-Trisubstituted Pyrroles N. P. Buu-Hoï, Richard Rips, and Charles Derappe pp 1357 - 1362; DOI: 10.1021/jm01241a028 |
Phenyl-bridged Analogs of Phenylbutazone Harman S. Lowrie pp 1362 - 1364; DOI: 10.1021/jm01241a029 |
Methanesulfonates of Tertiary and Quaternary Amino Alcohols Sara Ginsburg pp 1364 - 1367; DOI: 10.1021/jm01241a030 |
Aldehyde Hydrazone Derivatives in Cancer Chemotherapy Richard H. Wiley and R. L. Clevenger pp 1367 - 1371; DOI: 10.1021/jm01241a031 |
Penetration of Brain and Brain Tumors by Intravascular Injection of Alkylating Agents. IV Albert H. Soloway, Emery Nyilas, Raymond N. Kjellberg, and Vernon H. Mark pp 1371 - 1376; DOI: 10.1021/jm01241a032 |
Constituents of Cocculus Leaeba DC--Correction for Mistaken Botanical Identity A. V. Subbaratnam and William B. Cook pp 1376 - 1378; DOI: 10.1021/jm01241a033 |
Some 2-Substituted 2H-1,4-Benzoxazin-3(4H)-ones Keith W. Wheeler pp 1378 - 1383; DOI: 10.1021/jm01241a034 |
Book Reviews pp 1384 - 1384; DOI: 10.1021/jm01241a036 |
ERRATUM: Chemistry and Structure-Activity Relationships of Mecamylamine and Derivatives Clement A. Stone, Mary L. Torchiana, Meyer Sletzinger, Gustav A. Stein, William V. Ruyle, Donald F. Reinhold, Walter A. Gaines, Heinz Arnold, and Karl Pfister pp 1385 - 1385; DOI: 10.1021/jm01241a037 |